Missing Links?: 7650 Citation Matrix | Graphs | Glossary HistCite Guide About |
Nodes: 29221,
Authors: 40665,
Journals: 1485,
Outer References: 554040,
Words: 41910
Collection span: 1946 - 2005
View: Overview. Sorted by journal name.
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# | LCR | NCR | Node / Date / Journal / Author | LCS | GCS |
---|---|---|---|---|---|
12101 | 6 | 36 | 8479 1970 JOURNAL OF MEDICINAL CHEMISTRY 13 (3): 475-& SADEE W FRAGMENTATION PATTERN OF 1,4-BENZODIAZEPIN-2-ONES UNDER ELECTRON IMPACT | 5 | 39 |
12102 | 3 | 16 | 8480 1970 JOURNAL OF MEDICINAL CHEMISTRY 13 (3): 531-& WOLFF ME; ZANATI G; SHANMUGA.G; GUPTE S; AADAHL G THIA STEROIDS .3. DERIVATIVES OF 2-THIA-A-NOR-5ALPHA-ANDROSTAN-17BETA-OL AS PROBES OF STEROID-RECEPTOR INTERACTIONS | 0 | 14 |
12103 | 1 | 18 | 8481 1970 JOURNAL OF MEDICINAL CHEMISTRY 13 (3): 561-& GOLDKAMP AH CHLOROSULFONATION OF 17BETA-ACETOXY-3-METHOXYESTRA-1,3,5(10)-TRIENE | 0 | 1 |
12104 | 3 | 35 | 9462 1971 JOURNAL OF MEDICINAL CHEMISTRY 14 (1): 24-& WITIAK DT; MUHIELDE.Z; MAHISHI N; SETHI OP; GERALD MC L(S)- AND D(R)-3-AMINO-1-PHENYLPYRROLIDINES - STEREOSELECTIVE ANTAGONISTS FOR HISTAMINE AND ACETYLCHOLINE RECEPTORS IN-VITRO | 0 | 19 |
12105 | 1 | 18 | 9463 1971 JOURNAL OF MEDICINAL CHEMISTRY 14 (4): 331-& REMERS WA; GREENBLA.EN; ELLENBOG.L; WEISS MJ 5,8-DIHYDROHARMAN DERIVATIVES - THEIR PREPARATION AND BIOLOGICAL ACTIVITIES | 1 | 4 |
12106 | 3 | 7 | 9464 1971 JOURNAL OF MEDICINAL CHEMISTRY 14 (7): 629-& LEMAHIEU RA; BORIS A; CARSON M; KIERSTEA.RW SYNTHESIS OF SOME 3,7-DIHYDROXY-6-METHYL-DELTA5-PREGNENE DERIVATIVES | 1 | 2 |
12107 | 3 | 21 | 9465 1971 JOURNAL OF MEDICINAL CHEMISTRY 14 (12): 1178-& MCILHENN.HM METABOLISM OF [C-14]VERAPAMIL | 0 | 76 |
12108 | 4 | 19 | 9466 1971 JOURNAL OF MEDICINAL CHEMISTRY 14 (12): 1190-& BIOLLAZ M; LANDEROS RM; CUELLAR L; CRABBE P; ROOKS W; et al. 17 ALPHA-PROPADIENYL-19-NORTESTOSTERONE AND RELATED COMPOUNDS - NEW SERIES OF POTENT ORALLY ACTIVE PROGESTOGENS | 2 | 13 |
12109 | 2 | 12 | 10494 1972 JOURNAL OF MEDICINAL CHEMISTRY 15 (1): 89-& EADON G; DJERASSI C SYNTHESIS AND BIOLOGICAL-ACTIVITY OF D-BISHOMO STEROIDS | 1 | 1 |
12110 | 8 | 39 | 10495 1972 JOURNAL OF MEDICINAL CHEMISTRY 15 (4): 360-& JOHNSON AL (+/-)-6,6-DIFLUORONORGESTREL, A NEW SYNTHETIC HORMONAL STEROID | 0 | 8 |
# | LCR | NCR | Node / Date / Journal / Author | LCS | GCS |
12111 | 2 | 31 | 10496 1972 JOURNAL OF MEDICINAL CHEMISTRY 15 (4): 374-& WILEY RA; HAVA MM; FARAJ BA; JANTZ A INFLUENCE OF STEREOCHEMISTRY AND LIPOPHILICITY ON BIOLOGICAL-ACTIVITY OF SOME GANGLIONIC BLOCKING-AGENTS | 0 | 15 |
12112 | 0 | 25 | 10497 1972 JOURNAL OF MEDICINAL CHEMISTRY 15 (6): 615-& LIN AJ; SARTOREL.AC; AGRAWAL KC POTENTIAL ANTITUMOR AGENTS .8. DERIVATIVES OF 3-BENZYLOXY-2-FORMYLPYRIDINE AND 5-BENZYLOXY-2-FORMYLPYRIDINE THIOSEMICARBAZONE | 0 | 10 |
12113 | 3 | 13 | 10498 1972 JOURNAL OF MEDICINAL CHEMISTRY 15 (6): 679-& FARO HP; HERZOG HL; NERI R; YOUNGSTR.RE; POPPER TL PREPARATION AND PROGESTATIONAL ACTIVITY OF 6-TRIFLUOROMETHYL-16-METHYLENE-17 ALPHA-HYDROXY-4,6-PREGNADIENE-3,20-DIONE 17-ACETATE AND RELATED COMPOUNDS | 1 | 3 |
12114 | 4 | 18 | 10499 1972 JOURNAL OF MEDICINAL CHEMISTRY 15 (7): 784-& JOHNSON AL 6,6-DIFLUORO-19-NORPROGESTERONE | 0 | 1 |
12115 | 1 | 13 | 10500 1972 JOURNAL OF MEDICINAL CHEMISTRY 15 (8): 840-& DAGNE E; CASTAGNO.N COTININE N-OXIDE, A NEW METABOLITE OF NICOTINE | 4 | 40 |
12116 | 9 | 36 | 10501 1972 JOURNAL OF MEDICINAL CHEMISTRY 15 (9): 909-& VANDERSI.D; KOOREMAN HJ; JAITLY KD; MARX AF 14ALPHA,17ALPHA-ALKYLIDENEDIOXYPROGESTERONE DERIVATIVES | 0 | 5 |
12117 | 3 | 16 | 10502 1972 JOURNAL OF MEDICINAL CHEMISTRY 15 (10): 1056-& FAHRENHO.KE; MEYERS KP; KIERSTEA.RW CYCLOPROP[16ALPHA, 17ALPHA] ANDROSTANES | 0 | 2 |
12118 | 4 | 17 | 10503 1972 JOURNAL OF MEDICINAL CHEMISTRY 15 (11): 1165-& RASMUSSO.GH; REYNOLDS GF; CHEN A; ARTH GE; PATANELL.DJ; et al. ANTIANDROGENS 2',3'ALPHA-TETRAHYDROFURAN-2'-SPIRO-17-(1,2ALPHA-METHYLENE-4-ANDROSTEN-3-ONES) | 0 | 15 |
12119 | 4 | 11 | 11465 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (1): 30-33 BILLETS S; LIETMAN PS; FENSELAU C MASS-SPECTRAL ANALYSIS OF GLUCURONIDES | 12 | 91 |
12120 | 7 | 30 | 11466 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (2): 93-97 MITSCHER LA; HOWISON PW; LAPIDUS JB; SOKOLOSK.TD CIRCULAR-DICHROISM STUDIES OF ARYL DIASTEREOISOMERS .2. DEPENDENCE OF 1LB TRANSITION SIGN UPON NATURE OF PARA SUBSTITUENT IN VARIOUS CHLORAMPHENICOL DERIVATIVES | 2 | 13 |
# | LCR | NCR | Node / Date / Journal / Author | LCS | GCS |
12121 | 8 | 26 | 11467 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (3): 257-262 GUTHRIE RW; BORIS A; MULLIN JG; MENNONA FA; KIERSTEA.RW PREPARATION OF SOME 7-OXAANDROSTANE DERIVATIVES | 3 | 6 |
12122 | 2 | 18 | 11468 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (5): 516-519 SHTACHER G; EREZ M; COHEN S SELECTIVITY IN NEW BETA-ADRENERGIC BLOCKING-AGENTS - (3-AMINO-2-HYDROXYPROPOXY)BENZAMIDES | 1 | 20 |
12123 | 6 | 10 | 11469 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (5): 568-570 JOHNS WF; HOFMANN LM 7-ACETYLTHIOETIOJERVANES - NEW ANTIALDOSTERONE AGENTS | 0 | 1 |
12124 | 7 | 14 | 11470 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (6): 647-649 LEMAHIEU RA; BORIS A; CARSON M; GUTHRIE RW; KIERSTEA.RW PREPARATION OF 17ALPHA-ACETOXY-7-OXAPROGESTERONE | 1 | 2 |
12125 | 11 | 30 | 11471 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (6): 649-654 SHAPIRO EL; WEBER L; TEUTSCH G; HARRIS H; NERI R; et al. 19-NORPROGESTINS - SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 6-CHLORO-16-METHYLENE-17ALPHA-HYDROXY-19-NOR-4,6-PREGNADIENE-3,20-DIONE 17-ACETATE | 0 | 3 |
12126 | 1 | 24 | 11472 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (9): 996-1002 DUNN GL; GALLAGHE.G; DAVIS LD; HOOVER JRE METABOLITES OF METHYL "5(6)-BUTYL-2-BENZIMIDAZOLECARBAMATE (PARBENDAZOLE) - STRUCTURE AND SYNTHESIS | 0 | 13 |
12127 | 3 | 42 | 11473 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (10): 1106-1112 NELSON SD; BRECK GD; TRAGER WF IN-VIVO METABOLITE CONDENSATIONS - FORMATION OF N-1-ETHYL-2-METHYL-N-3- (2,6-DIMETHYLPHENYL)-4-IMIDAZOLIDINONE FROM REACTION OF A METABOLITE OF ALCOHOL WITH A METABOLITE OF LIDOCAINE | 1 | 32 |
12128 | 0 | 19 | 11474 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (11): 1272-1276 DURANT GJ; LOYNES JM; WRIGHT SHB POTENTIAL HISTAMINE H2-RECEPTOR ANTAGONISTS .1. AMINOETHYLIMIDAZO[1,2-A]PYRIDINES AND IMIDAZO[1,5-A]PYRIDINES | 2 | 19 |
12129 | 1 | 30 | 11475 1973 JOURNAL OF MEDICINAL CHEMISTRY 16 (12): 1330-1333 SOLOMONS E; SAM J 2-AMINOINDANS OF PHARMACOLOGICAL INTEREST | 1 | 5 |
12130 | 2 | 26 | 12395 1974 JOURNAL OF MEDICINAL CHEMISTRY 17 (1): 65-72 CARNMALM B; JACUPOVI.E; JOHANSSO.L; PAULIS TD; RAMSBY S; et al. ANTIDEPRESSANT AGENTS .1. CHEMISTRY AND PHARMACOLOGY OF AMINO-SUBSTITUTED SPIRO[5H-DIBENZO[A,D]CYCLOHEPTENE-5,1'-CYCLOALKANES] | 0 | 31 |
# | LCR | NCR | Node / Date / Journal / Author | LCS | GCS |
12131 | 1 | 18 | 12396 1974 JOURNAL OF MEDICINAL CHEMISTRY 17 (1): 124-129 HENKEL JG; BELL KH; PORTOGHE.PS STEREOCHEMICAL STUDIES ON MEDICINAL AGENTS .16. CONFORMATIONAL STUDIES OF METHADONE AND ISOMETHADONE UTILIZING CIRCULAR-DICHROISM AND PROTON MAGNETIC-RESONANCE | 0 | 19 |
12132 | 1 | 9 | 12397 1974 JOURNAL OF MEDICINAL CHEMISTRY 17 (6): 654-657 KALTENBR.JS; RHEE TO 4-(2-THIENYL)-1-NAPHTHALENEACETIC ACIDS AND 5-(2-THIENYL)-1-NAPHTHALENEACETIC ACIDS AS ANTIINFLAMMATORY AGENTS | 0 | 2 |
12133 | 1 | 32 | 12398 1974 JOURNAL OF MEDICINAL CHEMISTRY 17 (7): 702-708 BAILEY DM; DEGRAZIA CG; WOOD D; SIGGINS J AMINE FUNCTIONS OF REDUCED BASICITY - HYPOGLYCEMIC AND NATRIURETIC ALPHA-ALKOXYBENZYLAMIDOXIMES, AMIDINES, AND CYCLOAMIDINES | 0 | 7 |
12134 | 2 | 19 | 12399 1974 JOURNAL OF MEDICINAL CHEMISTRY 17 (12): 1330-1333 DAGNE E; GRUENKE L; CASTAGNO.N DEUTERIUM-ISOTOPE EFFECTS IN INVIVO METABOLISM OF COTININE | 4 | 19 |
12135 | 5 | 18 | 13356 1975 JOURNAL OF MEDICINAL CHEMISTRY 18 (3): 268-271 CHINN LJ; DESAI BN SYNTHESIS OF 15-KETO-6-BETA,7-BETA-METHYLENEPROGESTERONE - EFFECT OF 6-BETA,7-BETA-METHYLENE GROUP ON MINERALOCORTICOID ACTIVITY | 2 | 6 |
12136 | 2 | 44 | 13357 1975 JOURNAL OF MEDICINAL CHEMISTRY 18 (4): 376-383 TAKAMIZAWA A; MATSUMOTO S; IWATA T; TOCHINO Y; KATAGIRI K; et al. STUDIES ON CYCLOPHOSPHAMIDE METABOLITES AND THEIR RELATED COMPOUNDS .2. PREPARATION OF AN ACTIVE SPECIES OF CYCLOPHOSPHAMIDE AND RELATED COMPOUNDS | 0 | 79 |
12137 | 7 | 28 | 13358 1975 JOURNAL OF MEDICINAL CHEMISTRY 18 (11): 1143-1145 KANOJIA RM; OSTROWSKI P; HAHN DW; ALLEN G; MCGUIRE JL 17ALPHA-ETHYL-20ALPHA-DIHYDROPROGESTERONES AND 20BETA-DIHYDROPROGESTERONES AND OTHER 17 ALPHA-ETHYL-SUBSTITUTED PREGNANES AS POTENTIAL CONTRAGESTATIONAL AGENTS | 0 | 2 |
12138 | 4 | 61 | 14244 1976 JOURNAL OF MEDICINAL CHEMISTRY 19 (7): 892-898 KORNET MJ; THIO AP OXINDOLE-3-SPIROPYRROLIDINES AND OXINDOLE-3-PIPERIDINES - SYNTHESIS AND LOCAL-ANESTHETIC ACTIVITY | 0 | 34 |
12139 | 13 | 33 | 15068 1977 JOURNAL OF MEDICINAL CHEMISTRY 20 (2): 213-220 TOSCANO L; GRISANTI G; FIORIELLO G; BARLOTTI L; BIANCHETTI A; et al. SYNTHESIS AND TOPICAL ANTIINFLAMMATORY PROPERTIES OF 17,21-BIS(ACETYLOXY)-6BETA,9-DIFLUORO-11BETA-HYDROXYPREGNA-1,4-DIENE-3,20-DIONE AND RELATED 2-HALOGENATED COMPOUNDS | 2 | 9 |
12140 | 0 | 10 | 15069 1977 JOURNAL OF MEDICINAL CHEMISTRY 20 (5): 726-728 SPRAGUE PW; HEIKES JE SYNTHESIS AND ANTIINFLAMMATORY ACTIVITY OF CIS-4,5,6,7,8,8A,9-HEXAHYDRO-ALPHA-METHYL-5H-FLUORENE-2-ACETIC ACID | 0 | 2 |
# | LCR | NCR | Node / Date / Journal / Author | LCS | GCS |
12141 | 3 | 9 | 15070 1977 JOURNAL OF MEDICINAL CHEMISTRY 20 (8): 1096-1099 CLARK ER; OMAR AME; PRESTWICH G POTENTIAL STEROIDAL ANTIESTROGENS | 6 | 22 |
12142 | 2 | 18 | 15071 1977 JOURNAL OF MEDICINAL CHEMISTRY 20 (10): 1312-1317 ARCHER GA; KALISH RI; NING RY; SLUBOSKI BC; STEMPEL A; et al. QUINAZOLINES AND 1,4-BENZODIAZEPINES .82. 5-PYRIMIDYLBENZODIAZEPINES AND 5-PYRAZINYLBENZODIAZEPINES | 0 | 11 |
12143 | 5 | 29 | 15072 1977 JOURNAL OF MEDICINAL CHEMISTRY 20 (11): 1493-1496 CAVESTRI RC; MOKOTOFF M AZABICYCLO CHEMISTRY .6. INVESTIGATION OF ONE OF CHEMICAL PARAMETERS FOR ANALGETIC ACTIVITY - SYNTHESIS OF 2-METHYL-2-AZABICYCLO[3.3.1]NON-6-ENE AND 2-METHYL-2-AZABICYCLO[3.3.1]NON-7-ENE | 0 | 5 |
12144 | 0 | 11 | 15876 1978 JOURNAL OF MEDICINAL CHEMISTRY 21 (3): 284-288 GELBART A; THOMAS R CARDENOLIDE ANALOGS .7. SYNTHESIS AND BIOLOGICAL-ACTIVITY OF SOME NEW STEROIDAL GUANYLHYDRAZONES | 2 | 20 |
12145 | 4 | 35 | 15877 1978 JOURNAL OF MEDICINAL CHEMISTRY 21 (7): 683-686 TESTA B; MIHAILOVA D ABINITIO STUDY OF ELECTRONIC FACTORS IN METABOLIC HYDROXYLATION OF ALIPHATIC CARBON-ATOMS | 0 | 9 |
12146 | 5 | 27 | 15878 1978 JOURNAL OF MEDICINAL CHEMISTRY 21 (10): 1007-1011 BRUEGGEMEIER RW; FLOYD EE; COUNSELL RE SYNTHESIS AND BIOCHEMICAL EVALUATION OF INHIBITORS OF ESTROGEN BIOSYNTHESIS | 5 | 77 |
12147 | 6 | 28 | 16675 1979 JOURNAL OF MEDICINAL CHEMISTRY 22 (2): 129-133 SOLO AJ; KUMAR V; ALKS V; DUAX WL STRUCTURAL REQUIREMENTS FOR PROGESTATIONAL ACTIVITY - SYNTHESIS AND PROPERTIES OF RAC-8-ALPHA,9-BETA,10-ALPHA,14-BETA-PROGESTERONE | 1 | 2 |
12148 | 2 | 23 | 16676 1979 JOURNAL OF MEDICINAL CHEMISTRY 22 (4): 458-460 NICHOLS DE; WOODARD R; HATHAWAY BA; LOWY MT; YIM GKW RESOLUTION AND ABSOLUTE-CONFIGURATION OF TRANS-2-(2,5-DIMETHOXY-4-METHYLPHENYL)CYCLOPROPYLAMINE, A POTENT HALLUCINOGEN ANALOG | 1 | 12 |
12149 | 1 | 20 | 16677 1979 JOURNAL OF MEDICINAL CHEMISTRY 22 (6): 687-694 BALDWIN JJ; ENGELHARDT EL; HIRSCHMANN R; LUNDELL GF; PONTICELLO GS; et al. BETA-ADRENERGIC BLOCKING-AGENTS WITH ACUTE ANTIHYPERTENSIVE ACTIVITY | 0 | 21 |
12150 | 1 | 39 | 16678 1979 JOURNAL OF MEDICINAL CHEMISTRY 22 (11): 1340-1346 SCHAAF TK; HESS HJ SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CARBOXYL-TERMINUS MODIFIED PROSTAGLANDIN ANALOGS | 0 | 41 |
# | LCR | NCR | Node / Date / Journal / Author | LCS | GCS |
12151 | 6 | 22 | 17390 1980 JOURNAL OF MEDICINAL CHEMISTRY 23 (7): 722-726 KONOPELSKI JP; DJERASSI C; RAYNAUD JP SYNTHESIS AND BIOCHEMICAL SCREENING OF PHENYLSELENIUM-SUBSTITUTED STEROID-HORMONES | 5 | 5 |
12152 | 1 | 49 | 17391 1980 JOURNAL OF MEDICINAL CHEMISTRY 23 (7): 764-773 HIRAI K; ISHIBA T; SUGIMOTO H; SASAKURA K; FUJISHITA T; et al. BENZOPHENONE RELATED-COMPOUNDS .2. PEPTIDOAMINOBENZOPHENONES, A NOVEL CLASS OF RING-OPENED DERIVATIVES OF 1,4-BENZODIAZEPINES | 0 | 27 |
12153 | 2 | 11 | 17392 1980 JOURNAL OF MEDICINAL CHEMISTRY 23 (8): 960-962 VINCEK WC; MARTIN BR; ACETO MD; BOWMAN ER SYNTHESIS AND PRELIMINARY BINDING-STUDIES OF 4,4-DITRITIO-(-)-NICOTINE OF HIGH SPECIFIC ACTIVITY | 0 | 19 |
12154 | 1 | 23 | 18087 1981 JOURNAL OF MEDICINAL CHEMISTRY 24 (3): 251-256 QUINN FR; BEISLER JA QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS OF COLCHICINES AGAINST P388 LEUKEMIA IN MICE | 0 | 32 |
12155 | 1 | 24 | 18817 1982 JOURNAL OF MEDICINAL CHEMISTRY 25 (2): 109-113 EISTETTER K; WOLF HPO SYNTHESIS AND HYPOGLYCEMIC ACTIVITY OF PHENYLALKYLOXIRANECARBOXYLIC ACID-DERIVATIVES | 0 | 30 |
12156 | 2 | 13 | 18818 1982 JOURNAL OF MEDICINAL CHEMISTRY 25 (12): 1488-1492 SADEK SA; KESSLER WV; SHAW SM; ANDERSON JN; WOLF GC SELENIUM LABELING IN NUCLEAR-MEDICINE .2. D-RING SUBSTITUTED ESTROGENS | 1 | 4 |
12157 | 1 | 18 | 19477 1983 JOURNAL OF MEDICINAL CHEMISTRY 26 (1): 1-6 LIPINSKI CA BIOISOSTERIC DESIGN OF CONFORMATIONALLY RESTRICTED PYRIDYLTRIAZOLE HISTAMINE H2-RECEPTOR ANTAGONISTS | 0 | 22 |
12158 | 2 | 22 | 19478 1983 JOURNAL OF MEDICINAL CHEMISTRY 26 (3): 367-372 TRYBULSKI EJ; BENJAMIN L; VITONE S; WALSER A; FRYER RI 2-BENZAZEPINES .4. [1,2,3]TRIAZOLO[4,5-D][2]BENZAZEPINES AND DIBENZO[C,F][1,2,3]TRIAZOLO[3,4-A]AZEPINES - SYNTHESIS AND EVALUATION AS CENTRAL NERVOUS-SYSTEM AGENTS | 0 | 11 |
12159 | 1 | 29 | 19479 1983 JOURNAL OF MEDICINAL CHEMISTRY 26 (6): 832-838 HEALD SL; JEFFS PW; LAVIN TN; NAMBI P; LEFKOWITZ RJ; et al. SYNTHESIS OF I125 LABELED (+/-)-15-(4-AZIDOBENZYL)CARAZOLOL - A POTENT BETA-ADRENERGIC PHOTOAFFINITY PROBE | 0 | 16 |
12160 | 2 | 17 | 19480 1983 JOURNAL OF MEDICINAL CHEMISTRY 26 (9): 1320-1323 SURCOUF E; LEPICARD G; MORNON JP; OJASOO T; RAYNAUD JP ADDITIONAL CONFORMATIONAL DATA FOR THE MAPPING OF THE PROGESTIN BINDING-SITE - CRYSTAL-STRUCTURES OF 21-(PHENYLSELENO)PROGESTERONE AND "17-ALPHA-(PHENYLSELENO)PROGESTERONE | 2 | 9 |
# | LCR | NCR | Node / Date / Journal / Author | LCS | GCS |
12161 | 18 | 62 | 20226 1984 JOURNAL OF MEDICINAL CHEMISTRY 27 (6): 734-740 LOVETT JA; DARBY MV; COUNSELL RE SYNTHESIS AND EVALUATION OF 19-AZAANDROSTENEDIONE AND 19-AMINOANDROSTENEDIONE ANALOGS AS POTENTIAL AROMATASE INHIBITORS | 0 | 17 |
12162 | 0 | 23 | 20877 1985 JOURNAL OF MEDICINAL CHEMISTRY 28 (10): 1414-1422 DURANT GJ; GANELLIN CR; HILLS DW; MILES PD; PARSONS ME; et al. THE HISTAMINE H2-RECEPTOR AGONIST IMPROMIDINE - SYNTHESIS AND STRUCTURE ACTIVITY CONSIDERATIONS | 0 | 44 |
12163 | 2 | 25 | 20878 1985 JOURNAL OF MEDICINAL CHEMISTRY 28 (11): 1695-1699 HOYTE RM; ROSNER W; JOHNSON IS; ZIELINSKI J; HOCHBERG RB SYNTHESIS AND EVALUATION OF POTENTIAL RADIOLIGANDS FOR THE PROGESTERONE-RECEPTOR | 3 | 30 |
12164 | 5 | 28 | 21448 1986 JOURNAL OF MEDICINAL CHEMISTRY 29 (10): 1917-1921 BIFTU T; GAMBLE NF; DOEBBER T; HWANG SB; SHEN TY; et al. CONFORMATION AND ACTIVITY OF TETRAHYDROFURAN LIGNANS AND ANALOGS AS SPECIFIC PLATELET-ACTIVATING-FACTOR ANTAGONISTS | 3 | 57 |
12165 | 1 | 28 | 22035 1987 JOURNAL OF MEDICINAL CHEMISTRY 30 (1): 24-29 ALOUP JC; BOUCHAUDON J; FARGE D; JAMES C; DEREGNAUCOURT J; et al. SYNTHESIS AND ANTISECRETORY AND ANTIULCER ACTIVITIES OF DERIVATIVES AND ANALOGS OF 2-(2-PYRIDYL)TETRAHYDROTHIOPHENE-2-CARBOTHIOAMIDE | 0 | 19 |
12166 | 1 | 31 | 22036 1987 JOURNAL OF MEDICINAL CHEMISTRY 30 (2): 249-254 PETERSON LA; TREVOR A; CASTAGNOLI N STEREOCHEMICAL STUDIES ON THE CYTOCHROME-P-450 CATALYZED OXIDATION OF (S)-NICOTINE TO THE (S)-NICOTINE DELTA-1'(5')-IMINIUM SPECIES | 1 | 37 |
12167 | 7 | 19 | 22037 1987 JOURNAL OF MEDICINAL CHEMISTRY 30 (8): 1399-1403 LAM LKT; SPARNINS VL; WATTENBERG LW EFFECTS OF DERIVATIVES OF KAHWEOL AND CAFESTOL ON THE ACTIVITY OF GLUTATHIONE-S-TRANSFERASE IN MICE | 2 | 35 |
12168 | 1 | 34 | 22038 1987 JOURNAL OF MEDICINAL CHEMISTRY 30 (10): 1729-1737 BOLIS G; FUNG AKL; GREER J; KLEINERT HD; MARCOTTE PA; et al. RENIN INHIBITORS - DIPEPTIDE ANALOGS OF ANGIOTENSINOGEN INCORPORATING TRANSITION-STATE, NONPEPTIDIC REPLACEMENTS AT THE SCISSILE BOND | 1 | 37 |
12169 | 4 | 24 | 22545 1988 JOURNAL OF MEDICINAL CHEMISTRY 31 (3): 572-576 PETERS RH; CROWE DF; AVERY MA; CHONG WKM; TANABE M ANALOGS OF [(TRIETHYLSILYL)ETHYNYL]ESTRADIOL AS POTENTIAL ANTIFERTILITY AGENTS | 1 | 4 |
12170 | 2 | 23 | 22546 1988 JOURNAL OF MEDICINAL CHEMISTRY 31 (4): 730-736 PELLICCIARI R; NATALINI B; CECCHETTI S; PORTER B; RODA A; et al. BILE-ACIDS WITH A CYCLOPROPYL-CONTAINING SIDE-CHAIN .3. SEPARATION, IDENTIFICATION, AND PROPERTIES OF ALL 4 STEREOISOMERS OF 3-ALPHA,7-BETA-DIHYDROXY-22,23-METHYLENE-5-BETA-CHOLAN-24-OIC ACID | 0 | 11 |
# | LCR | NCR | Node / Date / Journal / Author | LCS | GCS |
12171 | 1 | 16 | 22547 1988 JOURNAL OF MEDICINAL CHEMISTRY 31 (5): 1005-1009 KELLEY JL; KROCHMAL MP; LINN JA; MCLEAN EW; SOROKO FE 9-(2-FLUOROBENZYL)-6-(ALKYLAMINO)-9H-PURINES - A NEW CLASS OF ANTICONVULSANT AGENTS | 0 | 20 |
12172 | 1 | 46 | 22548 1988 JOURNAL OF MEDICINAL CHEMISTRY 31 (9): 1729-1738 BORCHERDING DR; NARAYANAN S; HASOBE M; MCKEE JG; KELLER BT; et al. POTENTIAL INHIBITORS OF S-ADENOSYLMETHIONINE-DEPENDENT METHYLTRANSFERASES .11. MOLECULAR DISSECTIONS OF NEPLANOCIN-A AS POTENTIAL INHIBITORS OF S-ADENOSYLHOMOCYSTEINE HYDROLASE | 0 | 47 |
12173 | 2 | 12 | 22549 1988 JOURNAL OF MEDICINAL CHEMISTRY 31 (10): 1946-1950 ALI H; ROUSSEAU J; GHAFFARI MA; VANLIER JE SYNTHESIS, RECEPTOR-BINDING, AND TISSUE DISTRIBUTION OF (17-ALPHA,20E)- 21-[I-125]IODO-19-NORPREGNA-1,3,5(10),20-TETRAENE-3,17-DIOL AND (17-ALPHA,20Z)-21-[I-125]IODO-19-NORPREGNA-1,3,5(10),20-TETRAENE-3,17-DIOL | 1 | 41 |
12174 | 4 | 48 | 23102 1989 JOURNAL OF MEDICINAL CHEMISTRY 32 (3): 651-658 SHERWIN PF; MCMULLAN PC; COVEY DF EFFECTS OF STEROID D-RING MODIFICATION ON SUICIDE INACTIVATION AND COMPETITIVE-INHIBITION OF AROMATASE BY ANALOGS OF ANDROSTA-1,4-DIENE-3,17-DIONE | 2 | 20 |
12175 | 9 | 47 | 23103 1989 JOURNAL OF MEDICINAL CHEMISTRY 32 (7): 1642-1652 PETERS RH; CROWE DF; AVERY MA; CHONG WKM; TANABE M 17-DESOXY ESTROGEN ANALOGS | 3 | 19 |
12176 | 1 | 22 | 23610 1990 JOURNAL OF MEDICINAL CHEMISTRY 33 (4): 1246-1252 COOPER CS; KLOCK PL; CHU DTW; FERNANDES PB THE SYNTHESIS AND ANTIBACTERIAL ACTIVITIES OF QUINOLONES CONTAINING 5-MEMBERED AND 6-MEMBERED HETEROCYCLIC SUBSTITUENTS AT THE 7-POSITION | 0 | 9 |
12177 | 1 | 28 | 24107 1991 JOURNAL OF MEDICINAL CHEMISTRY 34 (8): 2402-2410 MOHAN R; CHOU YL; BIHOVSKY R; LUMMA WC; ERHARDT PW; et al. SYNTHESIS AND BIOLOGICAL-ACTIVITY OF ANGIOTENSIN-II ANALOGS CONTAINING A VAL-HIS REPLACEMENT, VAL-PSI[CH(CONH2)NH]HIS | 0 | 2 |
12178 | 1 | 44 | 25075 1993 JOURNAL OF MEDICINAL CHEMISTRY 36 (9): 1111-1119 KYM PR; CARLSON KE; KATZENELLENBOGEN JA PROGESTIN 16-ALPHA, 17-ALPHA-DIOXOLANE KETALS AS MOLECULAR PROBES FOR THE PROGESTERONE-RECEPTOR - SYNTHESIS, BINDING-AFFINITY, AND PHOTOCHEMICAL EVALUATION | 0 | 12 |
12179 | 1 | 72 | 25076 1993 JOURNAL OF MEDICINAL CHEMISTRY 36 (18): 2645-2657 CLARK RD; MILLER AB; BERGER J; REPKE DB; WEINHARDT KK; et al. 2-(QUINUCLIDIN-3-YL)PYRIDO[4,3-B]INDOL-1-ONES AND ISOQUINOLIN-1-ONES - POTENT CONFORMATIONALLY RESTRICTED 5-HT(3) RECEPTOR ANTAGONISTS | 1 | 41 |
12180 | 1 | 26 | 25077 1993 JOURNAL OF MEDICINAL CHEMISTRY 36 (22): 3361-3370 JOHNSON RE; BAIZMAN ER; BECKER C; BOHNET EA; BELL RH; et al. 4,5-DIHYDRO-1-PHENYL-1H-2,4-BENZODIAZEPINES - NOVEL ANTIARRHYTHMIC AGENTS | 0 | 8 |
# | LCR | NCR | Node / Date / Journal / Author | LCS | GCS |
12181 | 5 | 32 | 25078 1993 JOURNAL OF MEDICINAL CHEMISTRY 36 (24): 3956-3967 HU YF; ZORUMSKI CF; COVEY DF NEUROSTEROID ANALOGS - STRUCTURE-ACTIVITY STUDIES OF BENZ[E]INDENE MODULATORS OF GABA(A) RECEPTOR FUNCTION .1. THE EFFECT OF 6-METHYL SUBSTITUTION ON THE ELECTROPHYSIOLOGICAL ACTIVITY OF 7-SUBSTITUTED BENZ[E]INDENE-3-CARBONITRILES | 1 | 33 |
12182 | 1 | 44 | 25538 1994 JOURNAL OF MEDICINAL CHEMISTRY 37 (16): 2564-2573 FONTENLA JA; OSUNA J; ROSA E; CASTRO ME; GFERREIRO T; et al. SYNTHESIS AND ATYPICAL ANTIPSYCHOTIC PROFILE OF SOME 2-(2-PIPERIDINOETHYL)BENZOCYCLOALKANONES AS ANALOGS OF BUTYROPHENONE | 0 | 32 |
12183 | 1 | 21 | 25959 1995 JOURNAL OF MEDICINAL CHEMISTRY 38 (5): 771-793 BRESLIN HJ; KUKLA MJ; LUDOVICI DW; MOHRBACHER R; HO W; et al. SYNTHESIS AND ANTI-HIV-1 ACTIVITY OF 4,5,6,7-TETRAHYDRO-5-METHYLIMIDAZO[4,5,1-JK][1,4]BENZODIAZEPIN-2(1H)-ONE (TIBO) DERIVATIVES .3. | 0 | 43 |
12184 | 1 | 51 | 26340 1996 JOURNAL OF MEDICINAL CHEMISTRY 39 (1): 158-175 Jacobsen EJ; Tenbrink RE; Stelzer LS; Belonga KL; Carter DB; et al. High-affinity partial agonist imidazol[1,5-a]quinoxaline amides, carbamates, and ureas at the gamma-aminobutyric acid A benzodiazepine receptor complex | 0 | 31 |
12185 | 1 | 41 | 26341 1996 JOURNAL OF MEDICINAL CHEMISTRY 39 (15): 3001-3013 Zhang XY; Yao XT; Dalton JT; Shams G; Lei LP; et al. Medetomidine analogs as alpha 2-adrenergic ligands .2. Design, synthesis, and biological activity of conformationally restricted naphthalene derivatives of medetomidine | 0 | 7 |
12186 | 4 | 33 | 26712 1997 JOURNAL OF MEDICINAL CHEMISTRY 40 (20): 3297-3304 Ling YZ; Li JS; Liu Y; Kato K; Klus GT; et al. 17-imidazolyl, pyrazolyl, and isoxazolyl androstene derivatives. Novel steroidal inhibitors of human cytochrome C-17,C-20-lyase (P450(17 alpha)) | 1 | 43 |
12187 | 1 | 50 | 27110 1998 JOURNAL OF MEDICINAL CHEMISTRY 41 (3): 291-302 Zhi L; Tegley CM; Kallel EA; Marschke KB; Mais DE; et al. 5-aryl-1,2-dihydrochromeno[3,4-f]quinolines: A novel class of nonsteroidal human progesterone receptor agonists | 0 | 31 |
12188 | 1 | 43 | 27111 1998 JOURNAL OF MEDICINAL CHEMISTRY 41 (24): 4790-4799 Aronov AM; Verlinde CLMJ; Hol WGJ; Gelb MH Selective tight binding inhibitors of trypanosomal glyceraldehyde-3-phosphate dehydrogenase via structure-based drug design | 0 | 34 |
12189 | 7 | 48 | 27784 2000 JOURNAL OF MEDICINAL CHEMISTRY 43 (9): 1866-1877 Honda T; Gribble GW; Suh N; Finlay HJ; Rounds BV; et al. Novel synthetic oleanane and ursane triterpenoids with various enone functionalities in ring A as inhibitors of nitric oxide production in mouse macrophages | 0 | 18 |
12190 | 3 | 42 | 28360 2002 JOURNAL OF MEDICINAL CHEMISTRY 45 (1): 32-40 Gentili F; Bousquet P; Brasili L; Caretto M; Carrieri A; et al. alpha(2)-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole | 0 | 9 |
# | LCR | NCR | Node / Date / Journal / Author | LCS | GCS |
12191 | 2 | 31 | 28639 2003 JOURNAL OF MEDICINAL CHEMISTRY 46 (25): 5334-5348 Jiang X; Manion BD; Benz A; Rath NP; Evers AS; et al. Neurosteroid analogues. 9. Conformationally constrained pregnanes: Structure-activity studies of 13,24-cyclo-18,21-dinorcholane analogues of the GABA modulatory and anesthetic steroids (3 alpha,5 alpha)- and (3 alpha,5 beta)-3-hydroxypregnan-20-one | 0 | 3 |
12192 | 1 | 71 | 28640 2003 JOURNAL OF MEDICINAL CHEMISTRY 46 (26): 5812-5824 Govoni M; Bakker RA; van de Wetering I; Smit MJ; Menge WMBP; et al. Synthesis and pharmacological identification of neutral histamine H-1-receptor antagonists | 0 | 1 |
12193 | 3 | 21 | 28903 2004 JOURNAL OF MEDICINAL CHEMISTRY 47 (13): 3381-3387 Madauss KP; Deng SJ; Austin RJH; Lambert MH; McLay I; et al. Progesterone receptor ligand binding pocket flexibility: Crystal structures of the norethindrone and mometasone furoate complexes | 0 | 1 |
12194 | 1 | 25 | 29134 2005 JOURNAL OF MEDICINAL CHEMISTRY 48 (4): 1229-1236 Fecik RA; Devasthale P; Pillai S; Keschavarz-Shokri A; Shen L; et al. Chiral DNA gyrase inhibitors. 3. Probing the chiral preference of the active site of DNA gyrase. Synthesis of 10-fluoro-6-methyl-6,7-dihydro-9-piperazinyl-2H-benzo[a]quinolizin-20-one-3-carboxylic acid analogues | 0 | 0 |
12195 | 2 | 71 | 29135 2005 JOURNAL OF MEDICINAL CHEMISTRY 48 (14): 4628-4653 Thompson AM; Delaney AM; Hamby DM; Schroeder MC; Spoon TA; et al. Synthesis and structure-activity relationships of soluble 7-substituted 3-(3,5-dimethoxyphenyl)-1,6-naphthyridin-2-amines and related ureas as dual inhibitors of the fibroblast growth factor receptor-1 and vascular endothelial growth factor receptor-2 tyrosine kinases | 0 | 0 |
12196 | 0 | 26 | 27112 1998 JOURNAL OF MICROBIOLOGY AND BIOTECHNOLOGY 8 (6): 705-709 Ko HR; Kim BY; Ahn SC; Oh WK; Kim JH; et al. Chaetoglobosin A, an inhibitor of bleb formation on K562 cells induced by phorbol 12,13-dibutyrate | 0 | 1 |
12197 | 2 | 22 | 20227 1984 JOURNAL OF MICROSCOPY-OXFORD 134 (MAY): 221-224 FERRER JM; TATO A; STOCKERT JC BLUE MOLYBDENUM OXIDES - A STAIN FOR LIGHT AND ELECTRON-MICROSCOPY | 0 | 8 |
12198 | 1 | 45 | 29136 2005 JOURNAL OF MIDWIFERY & WOMENS HEALTH 50 (1): 31-38 Fehring RJ New low-and high-tech calendar methods of family planning | 0 | 0 |
12199 | 2 | 19 | 3356 1964 JOURNAL OF MOLECULAR BIOLOGY 8 (6): 863-& SAMEJIMA T; YANG JT OPTICAL ROTATORY DISPERSION OF SPERM-WHALE MYOGLOBIN + ITS DERIVATIVES | 11 | 62 |
12200 | 3 | 66 | 3357 1964 JOURNAL OF MOLECULAR BIOLOGY 10 (1): 73-& BRAHMS J; MOMMAERTS WFH STUDY OF CONFORMATION OF NUCLEIC ACIDS IN SOLUTION BY MEANS OF CIRCULAR DICHROISM | 9 | 253 |
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